5hes A 2.14 BS01 032 A 1 G23 F27 V30 A43 I66 I80 T82 E83 Y84 A85 C150 D151 F152 G153 G18 F22 V25 A38 I61 I75 T77 E78 Y79 A80 C145 D146 F147 G148 D133 K135 R137 N138 D151 T169 D128 K130 R132 N133 D146 T158 2.7.11.25 0004672,0005524,0006468 Kd=29nM -logKd/Ki=7.54, Kd=29nM IC50=23nM Q9NYL2 26999302 401 ASFVQIKFDDLQFFENCGGGSFGSVYRAKWISQDKEVAVKKLLKIEKEAEILSVLSHRNIIQFYGVILEPPNYGIVTEYASLGSLYDYINSNRSEEMDMDHIMTWATDVAKGMHYLHMEAPVKVIHRDLKSRNVVIAADGVLKICDFGASRFHNHTGTFPWMAPEVIQSLPVSETCDTYSYGVVLWEMLTREVPFKGLEGLQVAWLVVEKNERLTIPSSCPRSFAELLHQCWEADAKKRPSFKQIISILESMSNDTSLPDKCNSFLHNKAEWRCEIEATLERLKKLER 5hes B 2.14 BS01 032 B 1 G23 F27 V30 A43 K45 I66 T82 E83 Y84 A85 C150 D151 F152 G153 G17 F21 V24 A37 K39 I60 T76 E77 Y78 A79 C144 D145 F146 G147 D133 K135 R137 N138 D151 T169 D127 K129 R131 N132 D145 T149 2.7.11.25 0004672,0005524,0006468 Kd=29nM IC50=23nM Q9NYL2 26999302 401 SFVQIKFDDLQFFENCGGGSFGSVYRAKWISQDKEVAVKKLLKIEKEAEILSVLSHRNIIQFYGVILEPPNYGIVTEYASLGSLYDYINSNRSEEMDMDHIMTWATDVAKGMHYLHMEAPVKVIHRDLKSRNVVIAADGVLKICDFGGTFPWMAPEVIQSLPVSETCDTYSYGVVLWEMLTREVPFKGLEGLQVAWLVVEKNERLTIPSSCPRSFAELLHQCWEADAKKRPSFKQIISILESMSNDTSLPDKCNSFLHNKAEWRCEIEATLERLKKLE