5h8g A 2.0 BS01 5Y4 A 1 V53 V66 K68 I95 F113 V116 M163 I174 D175 V51 V64 K66 I91 F109 V112 M159 I170 D171 D156 K158 N161 D175 P184 S194 D152 K154 N157 D171 P180 S190 2.7.11.1 0004672,0004674,0005524,0006468 Kd=48.2pM -logKd/Ki=10.32, Kd=48.2pM IC50=<3.0nM, Kd=48nM P68400 26985319 421 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV