5h2u A 2.24 BS01 1N1 A 1 L197 A217 I218 K219 L248 I262 T264 M267 A268 G270 L319 G329 D330 L14 A34 I35 K36 L65 I79 T81 M84 A85 G87 L135 G145 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM -logKd/Ki=8.15, IC50=7nM Kd=7.8nM, IC50=5.3nM Q13882 27993680 501 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHHHH 5h2u B 2.24 BS01 1N1 B 1 L197 A217 I218 K219 L248 I262 T264 M267 A268 G270 D330 L14 A34 I35 K36 L65 I79 T81 M84 A85 G87 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM Kd=7.8nM, IC50=5.3nM Q13882 27993680 501 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHH 5h2u C 2.24 BS01 1N1 C 1 L197 A217 I218 K219 L248 I262 T264 M267 A268 K269 G270 E274 D330 L14 A34 I35 K36 L65 I79 T81 M84 A85 K86 G87 E91 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM Kd=7.8nM, IC50=5.3nM Q13882 27993680 501 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHHH 5h2u D 2.24 BS01 1N1 D 1 L197 A217 K219 L248 I262 T264 M267 A268 G270 L319 D330 L14 A34 K36 L65 I79 T81 M84 A85 G87 L135 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM Kd=7.8nM, IC50=5.3nM Q13882 27993680 504 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHH