5fd2 A 2.89 BS01 5XJ A 1 V471 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 V24 A34 K36 L58 L67 I80 T82 W84 C85 F136 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S160 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.05, IC50=90nM P15056 27085672 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 5fd2 B 2.89 BS01 5XJ B 1 V471 A481 K483 L514 W531 C532 D594 F595 V13 A23 K25 L45 W62 C63 D125 F126 D576 K578 N580 N581 D594 S616 D107 K109 N111 N112 D125 S130 2.7.11.1 0004672,0005524,0006468 P15056 27085672 801 DWEIPDGQITGTVYKGKWHGDVAVKMLAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS