5eyk A 1.93 BS01 peptide D 0 F117 I118 M119 R149 Y157 N158 Y226 K227 P352 P353 V354 Y355 F30 I31 M32 R62 Y70 N71 Y139 K140 P261 P262 V263 Y264 D216 K218 E220 N221 D234 T252 D129 K131 E133 N134 D147 T161 2.7.11.1 0004672,0005524,0006468 Q6DE08 27496137 805 ~ 826 FTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHARRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 5eyk A 1.93 BS02 5U5 A 1 L99 G100 K122 E141 Q145 L154 M156 L170 F172 A173 P174 G176 E177 L223 L12 G13 K35 E54 Q58 L67 M69 L83 F85 A86 P87 G89 E90 L136 D216 K218 E220 N221 D234 T252 D129 K131 E133 N134 D147 T161 2.7.11.1 0004672,0005524,0006468 ic50=3nM -logKd/Ki=8.52, IC50=3nM Q6DE08 27496137 401 FTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHARRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 5eyk B 1.93 BS01 5U5 B 1 L99 G100 K101 K122 E141 Q145 L154 L168 L170 F172 A173 G176 E177 L223 L19 G20 K21 K42 E61 Q65 L74 L88 L90 F92 A93 G96 E97 L143 D216 K218 E220 N221 D234 T252 D136 K138 E140 N141 D154 T172 2.7.11.1 0004672,0005524,0006468 ic50=3nM Q6DE08 27496137 401 AEMPKRKFTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQ