5ety A 2.9 BS01 ZN A 1 C1234 H1237 C1242 C1245 C130 H133 C138 C141 2.4.2.-,2.4.2.30 0003950 O95271 27196752 1401 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety A 2.9 BS02 K56 A 1 H1184 S1186 F1188 A1191 I1192 D1198 H1201 I1212 Y1213 Y1224 I1228 H80 S82 F84 A87 I88 D94 H97 I108 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 -logKd/Ki=7.51, IC50=31nM IC50=31nM O95271 27196752 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety B 2.9 BS01 ZN B 1 C1234 H1237 C1242 C1245 C127 H130 C135 C138 2.4.2.-,2.4.2.30 0003950 O95271 27196752 1401 GTILLDLAPEDKEYQSVEEEMQSTIREHGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety B 2.9 BS02 K56 B 1 H1184 S1186 F1188 A1191 I1192 D1198 H1201 I1212 Y1213 Y1224 I1228 H77 S79 F81 A84 I85 D91 H94 I105 Y106 Y117 I121 2.4.2.-,2.4.2.30 0003950 IC50=31nM O95271 27196752 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety C 2.9 BS01 ZN C 1 C1234 H1237 C1242 C1245 C127 H130 C135 C138 2.4.2.-,2.4.2.30 0003950 O95271 27196752 1401 GTILLDLAPEDKEYQSVEEEMQSTIREHRNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety C 2.9 BS02 K56 C 1 H1184 S1186 F1188 A1191 I1192 D1198 H1201 Y1213 H77 S79 F81 A84 I85 D91 H94 Y106 2.4.2.-,2.4.2.30 0003950 IC50=31nM O95271 27196752 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety D 2.9 BS01 ZN D 1 C1234 H1237 C1242 C1245 C128 H131 C136 C139 2.4.2.-,2.4.2.30 0003950 O95271 27196752 1401 GTILLDLAPEDKEYQSVEEEMQSTIREHRDNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE 5ety D 2.9 BS02 K56 D 1 S1186 F1188 A1191 I1192 D1198 H1201 Y1213 I1228 S80 F82 A85 I86 D92 H95 Y107 I122 2.4.2.-,2.4.2.30 0003950 IC50=31nM O95271 27196752 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPLAYAEYVIYRGEQAYPEYLITYQIMKPE