5e8z A 1.51 BS01 5L4 A 1 I211 G214 A230 K232 L260 Y282 H283 G286 L340 D351 I15 G18 A34 K36 L64 Y86 H87 G90 L144 D155 D333 K335 N338 D351 T375 D137 K139 N142 D155 T179 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=5.91, IC50=1.243uM P36897 27139629 601 GHMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE