5duf A 1.5 BS01 G7A A 1 L75 I76 H79 D83 Q103 D131 W133 L77 I78 H81 D85 Q105 D133 W135 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A62 D67 P74 I78 A102 Q105 P124 T125 L130 L132 D133 P212 W222 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 ic50=1.8uM -logKd/Ki=5.74, IC50=1.8uM P9WNP1 27571973 301 SHMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA