5acb C 2.7 BS01 5I1 C 1 I733 V741 A754 K756 F813 M816 D819 L866 Q1037 C1039 I18 V26 A39 K41 F98 M101 D104 L151 Q322 C324 D859 K861 S863 N864 D877 S889 T898 D144 K146 S148 N149 D162 S174 T183 2.7.11.22,2.7.11.23 0004672,0005524,0006468 -logKd/Ki=6.80, IC50=158nM Q9NYV4 27571479 2000 ESDWGKRCVDKFDIIGIIGEGTYGQVYKAKDKDTGELVALKKVRLDNEKEGFPITAIREIKILRQLIHRSVVNMKEIVTDKQDALDFKKDKGAFYLVFEYMDHDLMGLLESGLVHFSEDHIKSFMKQLMEGLEYCHKKNFLHRDIKCSNILLNNSGQIKLADFGLARLYNSEESRPYTNKVITLWYRPPELLLGEERYTPAIDVWSCGCILGELFTKKPIFQANLELAQLELISRLCGSPCPAVWPDVIKLPYFNTMKPKKQYRRRLREEFSFIPSAALDLLDHMLTLDPSKRCTAEQTLQSDFLKDVELSKMAPPDLPHWQDCH 5acb D 2.7 BS01 5I1 D 1 I733 V741 A754 K756 F813 M816 D819 E825 Q1037 C1039 E1041 I16 V24 A37 K39 F92 M95 D98 E104 Q313 C315 E317 D859 K861 S863 N864 D877 T898 D138 K140 S142 N143 D156 T174 2.7.11.22,2.7.11.23 0004672,0005524,0006468 Q9NYV4 27571479 2000 DWGKRCVDKFDIIGIIGEGTYGQVYKAKDKDTGELVALKKVRLDNEKEGFPITAIREIKILRQLIHRSVVNMKEIVTDKQFKKDKGAFYLVFEYMDHDLMGLLESGLVHFSEDHIKSFMKQLMEGLEYCHKKNFLHRDIKCSNILLNNSGQIKLADFGLARLYNSRPYTNKVITLWYRPPELLLGEERYTPAIDVWSCGCILGELFTKKPIFQANLELAQLELISRLCGSPCPAVWPDVIKLPYFNTMKPKKQYRRRLREEFSFIPSAALDLLDHMLTLDPSKRCTAEQTLQSDFLKDVELSKMAPPDLPHWQDCHELWS