5aaa A 1.73 BS01 VGH A 1 L1122 A1148 M1199 A1200 G1202 N1254 L1256 G1269 I1399 E1400 L30 A48 M99 A100 G102 N154 L156 G169 I293 E294 D1249 A1251 R1253 N1254 D1270 L1291 D149 A151 R153 N154 D170 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.38nM -logKd/Ki=9.42, Ki=0.38nM IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 26698910 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLEFMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE