4yv0 A 1.95 BS01 S4M A 1 L59 Q64 Y73 H74 G95 D98 D118 I119 G150 D168 T169 T170 L46 Q51 Y60 H61 G82 D85 D105 I106 G137 D155 T156 T157 2.5.1.16 0003824,0004766,0006596,0016740 Q4DA73 26327378 301 GWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 A 1.95 BS02 4JW B 1 E14 M24 L26 W53 P235 T236 E5 M11 L13 W40 P210 T211 2.5.1.16 0003824,0004766,0006596,0016740 -logKd/Ki=3.28, IC50=530uM Q4DA73 26327378 302 GWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 B 1.95 BS01 S4M B 1 Q40 L59 Q64 H74 G95 D98 D118 I119 D149 G150 D168 T169 T170 P175 A176 Q36 L55 Q60 H70 G91 D94 D114 I115 D145 G146 D164 T165 T166 P171 A172 2.5.1.16 0003824,0004766,0006596,0016740 Q4DA73 26327378 301 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 B 1.95 BS02 4JW B 1 E14 Q22 A23 M24 Y237 P238 C239 E10 Q18 A19 M20 Y233 P234 C235 2.5.1.16 0003824,0004766,0006596,0016740 ic50=530uM -logKd/Ki=3.28, IC50=530uM Q4DA73 26327378 302 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 C 1.95 BS01 S4M C 1 Q40 Q64 Y73 H74 G95 D98 D118 I119 G150 D168 T169 T170 Q30 Q54 Y63 H64 G85 D88 D108 I109 G140 D158 T159 T160 2.5.1.16 0003824,0004766,0006596,0016740 Q4DA73 26327378 301 ISGGWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 C 1.95 BS02 4JW D 1 M24 L26 P235 T236 M14 L16 P214 T215 2.5.1.16 0003824,0004766,0006596,0016740 Q4DA73 26327378 302 ISGGWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 D 1.95 BS01 S4M D 1 L59 Q64 Y73 H74 D98 D118 I119 D149 G150 D168 T169 T170 P175 L179 L55 Q60 Y69 H70 D94 D114 I115 D145 G146 D164 T165 T166 P171 L175 2.5.1.16 0003824,0004766,0006596,0016740 Q4DA73 26327378 301 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 D 1.95 BS02 4JW D 1 W19 Q22 A23 M24 Y237 P238 C239 W15 Q18 A19 M20 Y233 P234 C235 2.5.1.16 0003824,0004766,0006596,0016740 ic50=530uM Q4DA73 26327378 302 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN