4xv2 A 2.5 BS01 P06 A 1 G464 V471 A481 K483 L505 L514 F516 T529 W531 C532 F583 G593 D594 F595 G16 V23 A33 K35 L55 L64 F66 T79 W81 C82 F133 G143 D144 F145 D576 K578 N580 N581 D594 S616 D126 K128 N130 N131 D144 S148 2.7.11.1 0004672,0005524,0006468 ic50=0.00539uM -logKd/Ki=8.27, IC50=0.0054uM IC50=1.000000nM, EC50=529nM P15056 26466569 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 4xv2 B 2.5 BS01 P06 B 1 S465 V471 A481 K483 L505 L514 F516 T529 W531 C532 F583 G593 D594 F595 S18 V24 A34 K36 L58 L67 F69 T82 W84 C85 F134 G144 D145 F146 D576 K578 N580 N581 D594 S616 D127 K129 N131 N132 D145 S149 2.7.11.1 0004672,0005524,0006468 ic50=0.00539uM -logKd/Ki=8.27, IC50=0.0054uM IC50=1.000000nM, EC50=529nM P15056 26466569 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASEFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE