4xum A 2.4 BS01 IMN A 1 F282 C285 S289 H323 F360 F363 H449 Y473 F65 C68 S72 H106 F143 F146 H232 Y256 ? 0003677,0004879,0005634,0006355 ic50=21.3uM -logKd/Ki=4.67, IC50=21.3uM EC50=50000nM P37231 26445566 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xum A 2.4 BS02 IMN A 2 E259 R280 I281 C285 I341 S342 M348 E53 R63 I64 C68 I124 S125 M131 ? 0003677,0004879,0005634,0006355 ic50=21.3uM -logKd/Ki=4.67, IC50=21.3uM EC50=50000nM P37231 26445566 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xum B 2.4 BS01 IMN B 1 G284 C285 R288 I326 L333 I341 G67 C68 R71 I109 L116 I124 ? 0003677,0004879,0005634,0006355 ic50=21.3uM EC50=50000nM P37231 26445566 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGSPFVIYDMNSLMMGEDKIKFKHITPEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY