4wno A 1.56 BS01 3RF A 1 I22 V30 A44 M92 E93 Y94 C95 G98 L145 D165 I15 V23 A37 M85 E86 Y87 C88 G91 L138 D158 D138 K140 Q142 N143 D165 S184 D131 K133 Q135 N136 D158 S177 2.7.11.1 0004672,0004674,0005524,0006468,0010506 ic50=160nM -logKd/Ki=6.80, IC50=160nM O75385 25551253 401 TETVGKFEFSRKDLIGHGAFAVVFKGRHRAAHDLEVAVKCINKKNLAKSQTLLGKEIKILKELKHENIVALYDFQEMANSVYLVMEYCNGGDLADYLHAMRTLSEDTIRLFLQQIAGAMRLLHSKGIIHRDLKPQNILLSNPAGRRANPNSIRVKIADFGFARYLQSNMMAATLCGSPMYMAPEVIMSQHYDGKADLWSIGTIVYQCLTGKAPFQASSPQDLRLFYEKNKTLVPTIPRETSAPLRQLLLALLQRNHKDRMDFDEFFHHPFLDA