4v25 A 2.6 BS01 TF3 A 1 L63 P64 V67 G125 V126 Y129 N142 I143 F146 L56 P57 V60 G118 V119 Y122 N135 I136 F139 H239 E243 K246 N247 H225 E229 K232 N233 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0016310,0031670,0034614,0042593,0042803,0045254,0050848,0072332 IC50=2000nM Q15119 25404640 1367 GSAPKYIEHFSKFSPSPLSMKQFLDFGSACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTAPPLAGFGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVY 4v25 A 2.6 BS02 SZ6 A 1 K246 N247 R250 A251 D282 G284 G286 V287 T346 K232 N233 R236 A237 D268 G270 G272 V273 T323 H239 E243 K246 N247 H225 E229 K232 N233 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0016310,0031670,0034614,0042593,0042803,0045254,0050848,0072332 -logKd/Ki=7.08, IC50=84nM IC50=80nM Q15119 25404640 1369 GSAPKYIEHFSKFSPSPLSMKQFLDFGSACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTAPPLAGFGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVY