4v01 A 2.33 BS01 0LI A 1 A512 K514 E531 M534 M535 I545 V561 Y563 A564 I620 H621 L630 I639 A640 D641 A42 K44 E61 M64 M65 I75 V91 Y93 A94 I136 H137 L146 I155 A156 D157 D623 A625 R627 N628 D641 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 -logKd/Ki=8.11, Kd=7.7nM P11362 25465127 1776 LPEDPRWELPRDRLVLGKPLGGQVVLAEAIGLDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4v01 B 2.33 BS01 0LI B 1 A512 K514 E531 M534 V561 Y563 A564 I620 H621 L630 I639 A640 D641 F642 A47 K49 E66 M69 V96 Y98 A99 I140 H141 L150 I159 A160 D161 F162 D623 A625 R627 N628 D641 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005007,0005524,0006468 P11362 25465127 1770 SEYELPEDPRWELPRDRLVLGKPLGEGGQVVLAEAIGLDPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSN