4uy1 A 2.2 BS01 CA A 1 F26 G28 G30 D47 F26 G28 G30 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 O15496 25316315 200 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 4uy1 A 2.2 BS02 TJM A 1 L5 P17 Y20 G28 H46 D47 L5 P17 Y20 G28 H46 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=20uM -logKd/Ki=4.70, IC50=20uM IC50=20000nM O15496 25316315 1130 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 4uy1 B 2.2 BS01 CA B 1 F26 G28 G30 D47 F26 G28 G30 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 O15496 25316315 200 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD 4uy1 B 2.2 BS02 TJM B 1 L5 P17 F26 G28 H46 D47 L5 P17 F26 G28 H46 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=20uM IC50=20000nM O15496 25316315 1129 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD