4uxq A 1.85 BS01 0LI A 1 L473 V481 A501 K503 E520 M524 I527 I534 V550 A553 I609 H610 R611 L619 I628 A629 D630 F631 L22 V30 A50 K52 E69 M73 I76 I83 V99 A102 I145 H146 R147 L155 I164 A165 D166 F167 D612 A614 R616 N617 D630 D641 R650 D148 A150 R152 N153 D166 D177 R186 2.7.10.1 0004672,0004713,0005524,0006468 Kd=16nM -logKd/Ki=7.80, Kd=16.0nM IC50=8.0nM P22455 25465127 1752 LDLPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV