4ump A 2.3 BS01 5QM A 1 I17 A38 E57 L86 C89 L139 I149 I17 A38 E54 L83 C86 L136 I146 D132 K134 E136 N137 D150 A171 D129 K131 E133 N134 D147 A154 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 IC50=3100nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAGALAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4ump B 2.3 BS01 5QM B 1 I17 A38 E57 C89 I149 D150 I17 A38 E57 C89 I149 D150 D132 K134 E136 N137 D150 A171 D132 K134 E136 N137 D150 A165 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 IC50=3100nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKDCGALAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4ump C 2.3 BS01 5QM C 1 I17 V25 E57 L86 C89 L139 I149 I17 V22 E51 L80 C83 L133 I143 D132 K134 E136 N137 D150 A171 D126 K128 E130 N131 D144 A152 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 IC50=3100nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTAKVKLACHILTGEMVAIKIMDKNSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKGALAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4ump D 2.3 BS01 5QM D 1 A38 E57 L86 C89 L139 I149 A37 E56 L85 C88 L138 I148 D132 K134 E136 N137 D150 A171 D131 K133 E135 N136 D149 A163 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 IC50=3100nM Q14680 25589925 1334 KDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKDGALAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTISLWQYDHLTATYLLLLAKKARGKPVRLR