4ui4 A 2.4 BS01 ZN A 1 C1081 H1084 C1089 C1092 C130 H133 C138 C141 2.4.2.-,2.4.2.30 0003950 Q9H2K2 27163581 2115 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4ui4 A 2.4 BS02 RJN A 1 H1031 G1032 S1033 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 S82 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=45nM IC50=45nM Q9H2K2 27163581 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4ui4 B 2.4 BS01 ZN B 1 C1081 H1084 C1089 C1092 C130 H133 C138 C141 2.4.2.-,2.4.2.30 0003950 Q9H2K2 27163581 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4ui4 B 2.4 BS02 RJN B 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=45nM -logKd/Ki=7.35, IC50=45nM IC50=45nM Q9H2K2 27163581 2117 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM