4s3f A 1.7 BS01 43W A 1 M29 R56 D87 R110 R141 N145 K204 T231 R260 S262 M26 R53 D84 R107 R138 N142 K201 T228 R257 S259 1.17.7.3 0005506,0008299,0016114,0016491,0019288,0044237,0046429,0046872,0051539,0141197 ic50=580nM -logKd/Ki=6.24, IC50=580nM Q5SLI8 25868383 902 MRRPTPTVYVGRVPIGGAHPIAVQSMTNTPTRDVEATTAQVLELHRAGSEIVRLTVNDEEAAKAVPEIKRRLLAEGAEVPLVGDFHFNGHLLLRKYPKMAEALDKFRINPGTLGRGRHKDEHFAEMIRIAMDLGKPVRIGANWGSLDPALLTELMDRNARRPEPKSAHEVVLEALVESAVRAYEAALEMGLGEDKLVLSAKVSKARDLVWVYRELARRTQAPLHLGLTEAGMGVKGIVASAAALAPLLLEGIGDTIRVSLTPAPGEPRTKEVEVAQEILQALGLRAFAPEVTSCPGCGRTTSTFFQELAEEVSRRLKERLPEWRARYPGVEELKVAVMGCVVNGPGESKHAHIGISLPGAGEEPKAPVYADGKLLTILKGEGIAEEFLRLVEDYVKTRFAP