4rx8 A 1.59 BS01 3YX A 1 L377 A400 M448 M450 A451 G454 P455 R498 L501 S511 D512 L14 A37 M80 M82 A83 G86 P87 R130 L133 S143 D144 D494 A496 R498 N499 D512 K533 D126 A128 R130 N131 D144 K164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=35nM -logKd/Ki=7.46, IC50=35nM IC50=367nM, Kd=0.640000nM P43405 25633741 703 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHH