4rvl A 1.85 BS01 3XL A 1 L15 A36 K38 L84 E85 C87 G90 E91 L137 D148 L13 A28 K30 L69 E70 C72 G75 E76 L122 D133 D130 K132 E134 N135 D148 T170 D115 K117 E119 N120 D133 T155 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=41.7nM -logKd/Ki=7.38, IC50=41.7nM EC50=>5000nM, IC50=42nM O14757 25988399 301 VPFVEDWDLVQTLGVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA