4qrc A 1.901 BS01 0LI A 1 L473 A501 K503 E520 M524 V550 C552 A553 L603 C608 I609 H610 R611 L619 A629 D630 F631 L633 L20 A48 K50 E67 M71 V97 C99 A100 L150 C155 I156 H157 R158 L166 A176 D177 F178 L180 D612 A614 R616 N617 D630 R650 D159 A161 R163 N164 D177 R197 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.34, IC50=452nM IC50=8.0nM P22455 25317566 802 LPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPDLSPDGPRSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV