4qnu A 2.6 BS01 GEK A 1 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 -logKd/Ki=6.40, Kd=0.40uM A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQQHGLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu B 2.6 BS01 GEK B 1 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 K88 K107 G127 D149 P150 F154 I178 M193 G194 Y197 R312 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu C 2.6 BS01 GEK C 1 K91 K110 G130 D152 P153 F157 I181 E182 M196 G197 Y200 R315 K88 K107 G127 D149 P150 F154 I178 E179 M193 G194 Y197 R312 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu D 2.6 BS01 GEK D 1 K91 K110 G130 D152 P153 F157 G180 I181 M196 G197 Y200 R315 K91 K110 G130 D152 P153 F157 G180 I181 M196 G197 Y200 R315 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQQHGLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu E 2.6 BS01 GEK E 1 K91 W105 K110 G130 D152 P153 F157 G180 I181 M196 G197 Y200 R315 K87 W101 K106 G126 D148 P149 F153 G176 I177 M192 G193 Y196 R311 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu F 2.6 BS01 GEK F 1 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQQHGLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu G 2.6 BS01 GEK G 1 K91 W105 K110 G130 D152 P153 F157 G180 I181 E182 M196 G197 Y200 R315 K91 W105 K110 G130 D152 P153 F157 G180 I181 E182 M196 G197 Y200 R315 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQQHGLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qnu H 2.6 BS01 GEK H 1 K91 K110 G130 D152 P153 G180 I181 M196 Y200 R315 K88 K107 G127 D149 P150 G177 I178 M193 Y197 R312 2.5.1.- 0002098,0006400,0008033,0008168,0016740,0016765 A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP