4qfg A 3.46 BS01 STU A 1 L22 G23 G25 V30 A43 I77 M93 E94 Y95 V96 G99 E100 E143 N144 L146 D157 L14 G15 G17 V22 A35 I69 M85 E86 Y87 V88 G91 E92 E135 N136 L138 D149 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0000785,0002842,0003682,0004672,0004674,0004679,0005515,0005524,0005634,0005737,0005829,0006006,0006325,0006338,0006468,0006633,0006695,0006914,0008284,0008610,0009410,0009411,0009631,0010332,0010508,0010628,0010629,0014823,0016055,0016310,0016324,0016607,0017148,0019395,0030424,0030425,0031000,0031588,0031669,0032007,0032991,0033554,0034599,0042149,0042542,0042557,0042593,0042752,0043025,0043066,0043627,0044024,0044877,0045722,0045821,0045893,0046321,0046326,0046627,0046872,0047322,0048511,0048643,0050321,0050870,0050995,0055089,0060627,0061744,0061762,0062028,0070050,0070301,0070507,0071277,0071333,0071361,0071380,0071456,0071466,0097009,0106310,0140823,1903109,1903829,1903944,1903955,1904179,1904262,1904428,1905691,1990044,2000758 P54645 25066137 601 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFPWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDERPGSHTIEFFEMCANLIKILAQ 4qfg C 3.46 BS01 AMP C 1 H150 T199 I203 A204 V224 S225 I311 S313 S315 D316 H122 T171 I175 A176 V196 S197 I276 S278 S280 D281 ? 0004672,0004679,0005515,0005524,0005634,0005737,0005829,0006633,0010628,0016208,0019887,0019901,0031588,0031669,0032991,0043531,0044877,0051170 -logKd/Ki=5.48, Kd=3.3uM P80385 25066137 401 SSVYTTFMKSHRCYDLIPTSSKLVVFDTSLQVKKAFFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREVYLQPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFITEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDIYSKFDVINLAAEKTYNNLDVSVTKALQHRLKCYLHETLEAIINRLVEAEVHRLVVVDEHDVVKGIVSLSDILQALV