4q3t A 2.142 BS01 MN A 1 H131 D154 D158 D262 H106 D129 D133 D237 H131 D154 H156 D158 H171 D262 D264 E307 H106 D129 H131 D133 H146 D237 D239 E282 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 401 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3t A 2.142 BS02 MN A 2 D154 H156 D262 D264 D129 H131 D237 D239 H131 D154 H156 D158 H171 D262 D264 E307 H106 D129 H131 D133 H146 D237 D239 E282 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 402 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3t A 2.142 BS03 HAR A 1 D154 H156 D158 N160 H171 D213 D262 E307 D129 H131 D133 N135 H146 D188 D237 E282 H131 D154 H156 D158 H171 D262 D264 E307 H106 D129 H131 D133 H146 D237 D239 E282 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.33uM -logKd/Ki=6.48, Kd=0.33uM Q6WVP6 25007099 405 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3t B 2.142 BS01 MN B 1 H131 D154 D158 D262 H104 D127 D131 D235 H131 D154 H156 D158 H171 D262 D264 E307 H104 D127 H129 D131 H144 D235 D237 E280 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 401 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t B 2.142 BS02 MN B 2 D154 H156 D262 D264 D127 H129 D235 D237 H131 D154 H156 D158 H171 D262 D264 E307 H104 D127 H129 D131 H144 D235 D237 E280 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 402 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t B 2.142 BS03 HAR B 1 D154 H156 D158 N160 H171 G172 D213 D262 E307 D127 H129 D131 N133 H144 G145 D186 D235 E280 H131 D154 H156 D158 H171 D262 D264 E307 H104 D127 H129 D131 H144 D235 D237 E280 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.33uM Q6WVP6 25007099 405 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t C 2.142 BS01 MN C 1 H131 D154 D158 D262 H103 D126 D130 D234 H131 D154 H156 D158 H171 D262 D264 E307 H103 D126 H128 D130 H143 D234 D236 E279 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 401 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t C 2.142 BS02 MN C 2 D154 H156 D262 D264 D126 H128 D234 D236 H131 D154 H156 D158 H171 D262 D264 E307 H103 D126 H128 D130 H143 D234 D236 E279 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 402 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t C 2.142 BS03 HAR C 1 H131 H156 D158 N160 S167 H171 G172 D213 T276 E307 H103 H128 D130 N132 S139 H143 G144 D185 T248 E279 H131 D154 H156 D158 H171 D262 D264 E307 H103 D126 H128 D130 H143 D234 D236 E279 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.33uM Q6WVP6 25007099 405 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3t D 2.142 BS01 HAR D 1 D154 H156 D158 N160 S167 H171 D124 H126 D128 N130 S137 H141 H131 D154 H156 D158 H171 D262 D264 E307 H101 D124 H126 D128 H141 D232 D234 E277 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.33uM Q6WVP6 25007099 401 LLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAH 4q3t D 2.142 BS02 MN D 1 H131 D154 D158 D262 H101 D124 D128 D232 H131 D154 H156 D158 H171 D262 D264 E307 H101 D124 H126 D128 H141 D232 D234 E277 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 402 LLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAH 4q3t D 2.142 BS03 MN D 2 D154 H156 D262 D264 D124 H126 D232 D234 H131 D154 H156 D158 H171 D262 D264 E307 H101 D124 H126 D128 H141 D232 D234 E277 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Q6WVP6 25007099 403 LLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAH