4pgh A 2.8 BS01 SAM A 1 G206 D229 L230 D249 M250 K263 G198 D221 L222 D241 M242 K255 H267 D268 E296 E328 H259 D260 E288 E320 2.1.1.68 0005634,0005737,0006970,0007623,0008168,0008171,0008757,0009058,0009809,0010344,0010555,0017096,0030187,0030744,0030755,0031537,0032259,0033799,0042428,0046983,0047763,0048354,0051555,0090333 -logKd/Ki=4.89, Kd=13uM C5YH12 24948836 401 AAVADEEACMYAMQLASSSILPMTLKNALELGLLEVLQKDAGKALAAEEVVARLPVAPTNPAAADMVDRMLRLLASYDVVKCQMEDKDGKYERRYSAAPVGKWLTPNEDGVSMAALALMNQDKVLMESWYYLKDAVLDGGIPFNKAYGMTAFEYHGTDPRFNRVFNEGMKNHSVIITKKLLEFYTGFDESVSTLVDVGGGIGATLHAITSHHSHIRGVNFDLPHVISEAPPFPGVQHVGGDMFKSVPAGDAILMKWILHDWSDAHCATLLKNCYDALPEKGGKVIVVECVLPVTTDAVPKAQGVFHVDMIMLAHNPGGRERYEREFRDLAKAAGFSGFKATYIYANAWAIEFIK 4pgh B 2.8 BS01 SAM B 1 G206 D229 L230 D249 M250 F251 K263 I265 G201 D224 L225 D244 M245 F246 K258 I260 H267 D268 E296 E328 H262 D263 E291 E323 2.1.1.68 0005634,0005737,0006970,0007623,0008168,0008171,0008757,0009058,0009809,0010344,0010555,0017096,0030187,0030744,0030755,0031537,0032259,0033799,0042428,0046983,0047763,0048354,0051555,0090333 C5YH12 24948836 401 EDVAAVADEEACMYAMQLASSSILPMTLKNALELGLLEVLQKDAGKALAAEEVVARLPVAPTNPAAADMVDRMLRLLASYDVVKCQMEDKDGKYERRYSAAPVGKWLTPNEDGVSMAALALMNQDKVLMESWYYLKDAVLDGGIPFNKAYGMTAFEYHGTDPRFNRVFNEGMKNHSVIITKKLLEFYTGFDESVSTLVDVGGGIGATLHAITSHHSHIRGVNFDLPHVISEAPPFPGVQHVGGDMFKSVPAGDAILMKWILHDWSDAHCATLLKNCYDALPEKGGKVIVVECVLPVTTDAVPKAQGVFHVDMIMLAHNPGGRERYEREFRDLAKAAGFSGFKATYIYANAWAIEFIK 4pgh C 2.8 BS01 SAM C 1 G206 D229 L230 D249 M250 F251 K263 G197 D220 L221 D240 M241 F242 K254 H267 D268 E296 E328 H258 D259 E287 E319 2.1.1.68 0005634,0005737,0006970,0007623,0008168,0008171,0008757,0009058,0009809,0010344,0010555,0017096,0030187,0030744,0030755,0031537,0032259,0033799,0042428,0046983,0047763,0048354,0051555,0090333 C5YH12 24948836 401 AVADEEACMYAMQLASSSILPMTLKNALELGLLEVLQKDAGKALAAEEVVARLPVAPTNPAAADMVDRMLRLLASYDVVKCQMEDKDGKYERRYSAAPVGKWLTPNEDGVSMAALALMNQDKVLMESWYYLKDAVLDGGIPFNKAYGMTAFEYHGTDPRFNRVFNEGMKNHSVIITKKLLEFYTGFDESVSTLVDVGGGIGATLHAITSHHSHIRGVNFDLPHVISEAPPFPGVQHVGGDMFKSVPAGDAILMKWILHDWSDAHCATLLKNCYDALPEKGGKVIVVECVLPVTTDAVPKAQGVFHVDMIMLAHNPGGRERYEREFRDLAKAAGFSGFKATYIYANAWAIEFIK 4pgh D 2.8 BS01 SAM D 1 G206 D229 L230 D249 M250 K263 G202 D225 L226 D245 M246 K259 H267 D268 E296 E328 H263 D264 E292 E324 2.1.1.68 0005634,0005737,0006970,0007623,0008168,0008171,0008757,0009058,0009809,0010344,0010555,0017096,0030187,0030744,0030755,0031537,0032259,0033799,0042428,0046983,0047763,0048354,0051555,0090333 C5YH12 24948836 401 AEDVAAVADEEACMYAMQLASSSILPMTLKNALELGLLEVLQKDAGKALAAEEVVARLPVAPTNPAAADMVDRMLRLLASYDVVKCQMEDKDGKYERRYSAAPVGKWLTPNEDGVSMAALALMNQDKVLMESWYYLKDAVLDGGIPFNKAYGMTAFEYHGTDPRFNRVFNEGMKNHSVIITKKLLEFYTGFDESVSTLVDVGGGIGATLHAITSHHSHIRGVNFDLPHVISEAPPFPGVQHVGGDMFKSVPAGDAILMKWILHDWSDAHCATLLKNCYDALPEKGGKVIVVECVLPVTTDAVPKAQGVFHVDMIMLAHNPGGRERYEREFRDLAKAAGFSGFKATYIYANAWAIEFIK