4p7e A 2.4 BS01 2HB A 1 L855 G856 G861 S862 V863 A880 M929 Y931 L932 G935 L983 D994 L13 G14 G19 S20 V21 A38 M83 Y85 L86 G89 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=4.76, IC50=17.5uM IC50=>10000nM O60674 25369270 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG 4p7e B 2.4 BS01 2HB B 1 L855 G856 K857 G858 G861 A880 M929 Y931 L932 G935 L983 G993 D994 L16 G17 K18 G19 G22 A41 M86 Y88 L89 G92 L140 G150 D151 D976 A978 R980 N981 D994 S1016 D133 A135 R137 N138 D151 S173 2.7.10.2 0004672,0004713,0005524,0006468 IC50=>10000nM O60674 25369270 1201 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG