4ot6 A 2.05 BS01 2V1 A 1 L408 T410 V416 A428 M477 A478 G480 N484 L528 L15 T17 V23 A35 M84 A85 G87 N91 L135 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F166 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.92, IC50=1200nM Q06187 24712864 701 SWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE