4ojb A 2.0 BS01 198 A 1 L704 N705 Q711 M742 M745 V746 M749 F764 T877 M895 I899 L34 N35 Q41 M72 M75 V76 M79 F94 T199 M217 I221 ? IC50=248nM, Ki=509nM P10275 25091737 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSLMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT