4n9e A 1.72 BS01 2HL A 1 K189 H191 F193 R196 D219 V242 A244 S275 I309 R311 R349 I351 E376 N377 I378 A379 K173 H175 F177 R180 D203 V226 A228 S259 I293 R295 R333 I335 E360 N361 I362 A363 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM -logKd/Ki=7.82, IC50=0.015uM IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9e A 1.72 BS02 2HL B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM -logKd/Ki=7.82, IC50=0.015uM IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9e B 1.72 BS01 2HL A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM -logKd/Ki=7.82, IC50=0.015uM IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9e B 1.72 BS02 2HL B 1 K189 H191 F193 R196 D219 V242 A244 S275 I309 R311 R349 I351 E376 N377 I378 A379 K172 H174 F176 R179 D202 V225 A227 S258 I292 R294 R332 I334 E359 N360 I361 A362 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM -logKd/Ki=7.82, IC50=0.015uM IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL