4n98 A 1.7 BS01 4FC A 1 R152 Y154 T172 G174 R176 P242 V247 M362 R146 Y148 T166 G168 R170 P236 V241 M356 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=280uM -logKd/Ki=3.55, Ki=280uM P0A988 24592885 401 MKFTVEREHLLKPLQQVSGTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n98 A 1.7 BS02 CA A 1 G46 T47 E202 G40 T41 E196 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 P0A988 24592885 404 MKFTVEREHLLKPLQQVSGTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n98 A 1.7 BS03 CA A 2 S181 S356 S175 S350 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 P0A988 24592885 406 MKFTVEREHLLKPLQQVSGTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n98 A 1.7 BS04 CA A 3 V5 E6 H9 V5 E6 H9 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 P0A988 24592885 407 MKFTVEREHLLKPLQQVSGTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n98 B 1.7 BS01 CA B 1 G46 T47 E202 G39 T40 E195 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 P0A988 24592885 402 MKFTVEREHLLKPLQQVSGLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4n98 B 1.7 BS02 CA B 2 V5 E6 H9 V5 E6 H9 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 P0A988 24592885 405 MKFTVEREHLLKPLQQVSGLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL