4n1u A 1.6 BS01 2GE A 1 F27 N33 F72 F74 W117 D119 D120 F139 F25 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=5nM -logKd/Ki=8.30, IC50=5.0nM IC50=5.0nM, EC50=126nM P36639 24695224 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDT 4n1u B 1.6 BS01 2GE B 1 F27 N33 F72 F74 M81 W117 D119 D120 F139 F26 N32 F71 F73 M80 W116 D118 D119 F138 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=5nM IC50=5.0nM, EC50=126nM P36639 24695224 201 GASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDT