4mx9 A 3.1 BS01 2E8 A 1 V64 A77 K79 M111 L125 Y130 E134 D194 V23 A36 K38 M70 L84 Y89 E93 D153 D173 K175 E177 N178 D194 T213 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0004683,0005509,0005516,0005524,0005634,0005737,0006468,0009931,0016020,0016310,0018105,0035556,0046777,0046872 -logKd/Ki=8.59, IC50=2.6nM F0V9W9 24681759 601 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYYYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMKSMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSSELATIFGVSDVDSETWKNVLAEVDKNNDGEVDFDEFQQMLLKLCGN