4mr6 A 1.67 BS01 1K0 A 1 P371 F372 V376 L383 N429 H433 V435 P26 F27 V31 L38 N84 H88 V90 ? -logKd/Ki=6.60, Kd=251nM Kd=5800nM, IC50=251nM P25440 24248379 505 LSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD