4mq2	A	2.8	BS01	2C4	A	1	F170 K188 F238 M240 L241 S242 Y243 L294 V306 D307	F35 K53 F103 M105 L106 S107 Y108 L159 V171 D172	D287 K289 N292 D307 S324	D152 K154 N157 D172 S189	2.7.11.23,2.7.12.1	0004672,0004712,0005524,0006468,0046777			-logKd/Ki=7.01, IC50=0.097uM	IC50=97nM	Q13627	24239188	501 	YNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK
4mq2	B	2.8	BS01	2C4	B	1	K188 F238 M240 L241 Y243 V306 D307	K54 F102 M104 L105 Y107 V170 D171	D287 K289 N292 D307 S324	D151 K153 N156 D171 S188	2.7.11.23,2.7.12.1	0004672,0004712,0005524,0006468,0046777				IC50=97nM	Q13627	24239188	501 	VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK
4mq2	C	2.8	BS01	2C4	C	1	I165 F170 V173 F238 M240 L241 S242 L294 V306 D307	I31 F36 V39 F102 M104 L105 S106 L158 V170 D171	D287 K289 N292 D307 S324	D151 K153 N156 D171 S188	2.7.11.23,2.7.12.1	0004672,0004712,0005524,0006468,0046777				IC50=97nM	Q13627	24239188	501 	VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDGKREYKPPGTRKLHNILGVETGGPGGRRGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK
4mq2	D	2.8	BS01	2C4	D	1	I165 F170 K188 F238 L241 S242 Y243 L294 V306 D307	I31 F36 K54 F104 L107 S108 Y109 L160 V172 D173	D287 K289 N292 D307 S324	D153 K155 N158 D173 S190	2.7.11.23,2.7.12.1	0004672,0004712,0005524,0006468,0046777				IC50=97nM	Q13627	24239188	501 	VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKWNLKKTKKREYKPPGTRKLHNILGVETGGPHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK