4lng B 1.905 BS01 ZN B 1 D365 C367 H433 D297 C299 H360 H311 R359 K362 D365 C367 Y368 D423 D430 H433 H243 R291 K294 D297 C299 Y300 D350 D357 H360 2.5.1.58 0003824,0004659,0004660,0005965,0008270,0008318,0016853,0018343,0046872,0097354 Q4WPS9 24347326 601 HPGIPALFREPPLIHDLLSTETTELQSETVNKCLPLLKGIHNSQKGPFNKYGIPALQRKDHLEYLYDSLEDYPASFVALDASRPWMVYWALAGLCLLGEDVTRFRERVISTFTAAQNSTGGIGGGHGQMSHVASSYAAVLSIAMVGGEEAFKLIDRKAMWKWLGKLKQPDGGFTVCEGGEEDVRGAYCAMVVHALLDLPLALPPEAEARQNGLETFTDGLPEYLSRCQTYEGGISGSPGSEAHGAYAFCALACLCLLGRPEVVVPRYMNIATLLPWLSARQYAPEGGFSGRTNKLVDGCYSHWVGNCWPLVQAALDGTQPLSSVGNLYSREGLTRYILSCCQCKLGGLRDKPGKHPDSYHTCYALTGLSTVQYYHYCTDSSVSSKDDFSSAFSWKHDPNFASDGQGSDIGVFTENDRLVPFHPIFVIPHKSAEDIRVWFENQSFDL 4lng B 1.905 BS02 JAN B 1 W157 D365 C367 D430 Y432 H433 W89 D297 C299 D357 Y359 H360 H311 R359 K362 D365 C367 Y368 D423 D430 H433 H243 R291 K294 D297 C299 Y300 D350 D357 H360 2.5.1.58 0003824,0004659,0004660,0005965,0008270,0008318,0016853,0018343,0046872,0097354 -logKd/Ki=5.62, IC50=2400nM Q4WPS9 24347326 602 HPGIPALFREPPLIHDLLSTETTELQSETVNKCLPLLKGIHNSQKGPFNKYGIPALQRKDHLEYLYDSLEDYPASFVALDASRPWMVYWALAGLCLLGEDVTRFRERVISTFTAAQNSTGGIGGGHGQMSHVASSYAAVLSIAMVGGEEAFKLIDRKAMWKWLGKLKQPDGGFTVCEGGEEDVRGAYCAMVVHALLDLPLALPPEAEARQNGLETFTDGLPEYLSRCQTYEGGISGSPGSEAHGAYAFCALACLCLLGRPEVVVPRYMNIATLLPWLSARQYAPEGGFSGRTNKLVDGCYSHWVGNCWPLVQAALDGTQPLSSVGNLYSREGLTRYILSCCQCKLGGLRDKPGKHPDSYHTCYALTGLSTVQYYHYCTDSSVSSKDDFSSAFSWKHDPNFASDGQGSDIGVFTENDRLVPFHPIFVIPHKSAEDIRVWFENQSFDL 4lng B 1.905 BS03 FPP B 1 R252 H311 R359 K362 Y368 W371 R184 H243 R291 K294 Y300 W303 H311 R359 K362 D365 C367 Y368 D423 D430 H433 H243 R291 K294 D297 C299 Y300 D350 D357 H360 2.5.1.58 0003824,0004659,0004660,0005965,0008270,0008318,0016853,0018343,0046872,0097354 Q4WPS9 24347326 603 HPGIPALFREPPLIHDLLSTETTELQSETVNKCLPLLKGIHNSQKGPFNKYGIPALQRKDHLEYLYDSLEDYPASFVALDASRPWMVYWALAGLCLLGEDVTRFRERVISTFTAAQNSTGGIGGGHGQMSHVASSYAAVLSIAMVGGEEAFKLIDRKAMWKWLGKLKQPDGGFTVCEGGEEDVRGAYCAMVVHALLDLPLALPPEAEARQNGLETFTDGLPEYLSRCQTYEGGISGSPGSEAHGAYAFCALACLCLLGRPEVVVPRYMNIATLLPWLSARQYAPEGGFSGRTNKLVDGCYSHWVGNCWPLVQAALDGTQPLSSVGNLYSREGLTRYILSCCQCKLGGLRDKPGKHPDSYHTCYALTGLSTVQYYHYCTDSSVSSKDDFSSAFSWKHDPNFASDGQGSDIGVFTENDRLVPFHPIFVIPHKSAEDIRVWFENQSFDL