4l46 A 3.01 BS01 5FI A 1 Y79 G80 V82 A98 L102 Y151 L152 M202 T212 K218 F359 Y23 G24 V26 A42 L46 Y95 L96 M146 T156 K162 F296 D195 K197 E199 N200 D213 T233 D139 K141 E143 N144 D157 T173 2.7.11.1 0004672,0004674,0005524,0006468 Ki=20nM, IC50=160nM P23443 23731517 401 NRGPEKIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLEEDVSQFDSKFTRQTPVQVFLGFTYVAPS 4l46 A 3.01 BS02 ZN A 1 H222 H228 C231 H166 H168 C171 D195 K197 E199 N200 D213 T233 D139 K141 E143 N144 D157 T173 2.7.11.1 0004672,0004674,0005524,0006468 P23443 23731517 403 NRGPEKIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLEEDVSQFDSKFTRQTPVQVFLGFTYVAPS