4k4e A 2.3 BS01 ZN A 1 C1234 H1237 C1242 C1245 C131 H134 C139 C142 2.4.2.-,2.4.2.30 0003950 O95271 23701517 1401 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSAYAEYVIYRGEQAYPEYLITYQIMKPEH 4k4e A 2.3 BS02 K4E A 1 H1184 S1186 F1188 I1192 F1197 D1198 H1201 Y1203 I1212 Y1213 Y1224 G1227 H81 S83 F85 I89 F94 D95 H98 Y100 I109 Y110 Y121 G124 2.4.2.-,2.4.2.30 0003950 -logKd/Ki=7.62, IC50=24nM O95271 23701517 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSAYAEYVIYRGEQAYPEYLITYQIMKPEH 4k4e B 2.3 BS01 ZN B 1 C1234 H1237 C1242 C1245 C131 H134 C139 C142 2.4.2.-,2.4.2.30 0003950 O95271 23701517 1401 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPGHHSVIGRPYAEYVIYRGEQAYPEYLITYQIMKPEH 4k4e B 2.3 BS02 K4E B 1 F1188 A1191 F1197 D1198 H1201 I1212 Y1213 Y1224 G1227 F85 A88 F94 D95 H98 I109 Y110 Y121 G124 2.4.2.-,2.4.2.30 0003950 O95271 23701517 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPGHHSVIGRPYAEYVIYRGEQAYPEYLITYQIMKPEH