4igr A 2.65 BS01 3ZA A 1 Y491 P518 T520 R525 G690 A691 T692 E739 Y765 Y59 P86 T88 R93 G138 A139 T140 E187 Y213 ? 0015276,0016020 -logKd/Ki=7.20, Kd=63nM Ki=123nM P42264 23414088 901 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGC