4i0r A 2.1 BS01 1B4 A 1 A400 M448 M450 A451 E452 G454 P455 L501 A34 M77 M79 A80 E81 G83 P84 L130 D494 A496 R498 N499 D512 K533 D123 A125 R127 N128 D141 K158 2.7.10.2 0004672,0004713,0005524,0006468 ic50=14nM -logKd/Ki=7.85, IC50=14nM IC50=190nM P43405 23350847 701 VYLDRKLLTLEDELGSGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH