4h3x A 1.764 BS01 ZN A 1 H226 H230 H236 H121 H125 H131 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 301 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS02 ZN A 2 H175 D177 H190 H203 H70 D72 H85 H98 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 302 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS03 CA A 1 D182 G183 D185 L187 D205 E208 D77 G78 D80 L82 D100 E103 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 303 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS04 CA A 2 D131 D206 E208 D26 D101 E103 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 304 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS05 CA A 3 D165 G197 Q199 D201 D60 G92 Q94 D96 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 305 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS06 10B A 1 L187 L188 A189 L222 H226 E227 H230 H236 L243 Y245 M247 L82 L83 A84 L117 H121 E122 H125 H131 L138 Y140 M142 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 IC50=200nM P14780 23567804 306 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x A 1.764 BS07 10B B 1 Y245 P246 Y140 P141 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 IC50=200nM P14780 23567804 306 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS01 10B A 1 Y245 P246 Y140 P141 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 IC50=200nM P14780 23567804 306 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS02 ZN B 1 H226 H230 H236 H121 H125 H131 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 301 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS03 ZN B 2 H175 D177 H190 H203 H70 D72 H85 H98 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 302 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS04 CA B 1 D182 G183 D185 L187 D205 E208 D77 G78 D80 L82 D100 E103 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 303 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS05 CA B 2 D131 D206 E208 D26 D101 E103 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 304 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS06 CA B 3 D165 G197 Q199 D201 D60 G92 Q94 D96 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 305 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h3x B 1.764 BS07 10B B 1 L187 A189 L222 H226 E227 H230 H236 L243 Y245 M247 Y248 L82 A84 L117 H121 E122 H125 H131 L138 Y140 M142 Y143 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 IC50=200nM P14780 23567804 306 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG