4gdy A 2.89 BS01 0X1 A 1 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 G109 S110 Q111 Y135 N195 D223 P225 S253 S255 R263 R386 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 -logKd/Ki=7.08, IC50=84nM Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy A 2.89 BS02 0X1 B 1 R20 G39 Y74 S75 L293 R20 G32 Y67 S68 L286 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 -logKd/Ki=7.08, IC50=84nM Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy B 2.89 BS01 0X1 A 1 I19 M33 G39 Y74 S75 I19 M33 G39 Y74 S75 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 -logKd/Ki=7.08, IC50=84nM Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy B 2.89 BS02 0X1 B 1 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 -logKd/Ki=7.08, IC50=84nM Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP