4g2f A 1.699 BS01 C07 A 1 A651 K653 E670 T699 E700 M702 L753 S763 D764 A43 K45 E62 T91 E92 M94 L145 S155 D156 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.80, IC50=0.16uM P29320 24900387 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFGLSRVLPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRNPGSLKIITPSNLLL