4g19 A 2.0 BS01 GSH A 1 S22 N24 Y46 H70 T72 L73 D87 S88 Y148 R153 S21 N23 Y45 H69 T71 L72 D86 S87 Y147 R152 ? 0016740 ic50=261.5uM -logKd/Ki=3.58, IC50=261.5uM I6ZUH3 23007392 302 AQPIVFYDIPSNERIKHSPWSPNTWKIRYALNYKGLKYKTEWVEYPDIAGVVQKLGGKPTEKTPDGRDHYTLPVIYDPNTKKVVEDSAAIAKYLDETYPDTPKLFPAGTDAFQAAFLDFAWPVLGFPVFMLVILDTANSLLPRSHDYFRSTREQKFGKKLEELATEEEWAKVEAGLAKLKGYLDANGKGNDLLLMGAQGGITYSDIQIASFFVWAKIIWGEGSEKWKRLISLHDGKWAQFYAQFTKFEQVD 4g19 B 2.0 BS01 GSH B 1 S22 N24 Y46 H70 T72 L73 D87 S88 Y148 R153 S21 N23 Y45 H69 T71 L72 D86 S87 Y147 R152 ? 0016740 ic50=261.5uM I6ZUH3 23007392 302 AQPIVFYDIPSNERIKHSPWSPNTWKIRYALNYKGLKYKTEWVEYPDIAGVVQKLGGKPTEKTPDGRDHYTLPVIYDPNTKKVVEDSAAIAKYLDETYPDTPKLFPAGTDAFQAAFLDFAWPVLGFPVFMLVILDTANSLLPRSHDYFRSTREQKFGKKLEELATEEEWAKVEAGLAKLKGYLDANGKGNDLLLMGAQGGITYSDIQIASFFVWAKIIWGEGSEKWKRLISLHDGKWAQFYAQFTKFEQV 4g19 C 2.0 BS01 GSH C 1 S22 N24 H70 T72 L73 D87 S88 Y148 R153 S21 N23 H69 T71 L72 D86 S87 Y147 R152 ? 0016740 ic50=261.5uM I6ZUH3 23007392 302 AQPIVFYDIPSNERIKHSPWSPNTWKIRYALNYKGLKYKTEWVEYPDIAGVVQKLGGKPTEKTPDGRDHYTLPVIYDPNTKKVVEDSAAIAKYLDETYPDTPKLFPAGTDAFQAAFLDFAWPVLGFPVFMLVILDTANSLLPRSHDYFRSTREQKFGKKLEELATEEEWAKVEAGLAKLKGYLDANGKGNDLLLMGAQGGITYSDIQIASFFVWAKIIWGEGSEKWKRLISLHDGKWAQFYAQFTKFEQV 4g19 D 2.0 BS01 GSH D 1 S22 N24 Y46 H70 T72 L73 D87 S88 Y148 R153 S21 N23 Y45 H69 T71 L72 D86 S87 Y147 R152 ? 0016740 ic50=261.5uM I6ZUH3 23007392 303 AQPIVFYDIPSNERIKHSPWSPNTWKIRYALNYKGLKYKTEWVEYPDIAGVVQKLGGKPTEKTPDGRDHYTLPVIYDPNTKKVVEDSAAIAKYLDETYPDTPKLFPAGTDAFQAAFLDFAWPVLGFPVFMLVILDTANSLLPRSHDYFRSTREQKFGKKLEELATEEEWAKVEAGLAKLKGYLDANGKGNDLLLMGAQGGITYSDIQIASFFVWAKIIWGEGSEKWKRLISLHDGKWAQFYAQFTKFEQVD