4fgz A 1.994 BS01 CQA A 1 I30 F31 G32 G39 E42 L213 V216 E217 Y220 I22 F23 G24 G31 E34 L205 V208 E209 Y212 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM -logKd/Ki=2.87, IC50=1350uM IC50=1350000nM Q8IDQ9 22771008 301 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz A 1.994 BS02 CQA A 2 E171 Y175 G243 R246 K247 E163 Y167 G235 R238 K239 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM -logKd/Ki=2.87, IC50=1350uM IC50=1350000nM Q8IDQ9 22771008 302 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz A 1.994 BS03 SAH A 1 Y19 I36 S37 G63 D85 I86 D110 I111 R127 D128 A129 H132 Y11 I28 S29 G55 D77 I78 D102 I103 R119 D120 A121 H124 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Q8IDQ9 22771008 303 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz B 1.994 BS01 CQA B 1 I30 F31 G32 G39 E42 L213 V216 E217 Y220 I22 F23 G24 G31 E34 L205 V208 E209 Y212 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM IC50=1350000nM Q8IDQ9 22771008 301 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz B 1.994 BS02 CQA B 2 E171 E174 Y175 G243 R246 K247 E163 E166 Y167 G235 R238 K239 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM IC50=1350000nM Q8IDQ9 22771008 302 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz B 1.994 BS03 SAH B 1 Y19 I36 S37 G63 D85 I86 I111 R127 A129 H132 Y11 I28 S29 G55 D77 I78 I103 R119 A121 H124 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Q8IDQ9 22771008 303 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN