4f6u A 2.1 BS01 0SR A 1 Y32 A50 S62 R65 E66 I79 F97 A100 I171 A172 D173 Y34 A52 S64 R67 E68 I81 F99 A102 I168 A169 D170 D151 K153 N156 D173 T196 D148 K150 N153 D170 T176 2.7.11.22,2.7.11.23 0004672,0005524,0006468 -logKd/Ki=6.15, Kd=0.70uM P49336 23630251 501 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQENPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL