4ee0 A 1.75 BS01 0O4 A 1 F9 M11 G13 R14 D96 M99 W104 F8 M10 G12 R13 D91 M94 W99 Y8 R14 R19 W104 Y7 R13 R18 W99 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 -logKd/Ki=8.63, IC50=2.34nM IC50=2.34nM O60760 22546671 202 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4ee0 A 1.75 BS02 GSF A 1 Y8 R14 K50 I51 Q63 S64 Y7 R13 K45 I46 Q58 S59 Y8 R14 R19 W104 Y7 R13 R18 W99 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 O60760 22546671 203 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4ee0 B 1.75 BS01 0O4 B 1 F9 M11 G13 R14 D96 M99 S100 W104 F9 M11 G13 R14 D94 M97 S98 W102 Y8 R14 R19 W104 Y8 R14 R19 W102 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 IC50=2.34nM O60760 22546671 201 HPNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4ee0 B 1.75 BS02 GSF B 1 Y8 F9 R14 W39 K43 K50 I51 Q63 S64 Y8 F9 R14 W37 K41 K48 I49 Q61 S62 Y8 R14 R19 W104 Y8 R14 R19 W102 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 O60760 22546671 202 HPNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL