4e7r G 2.25 BS01 peptide M 0 E1023 I1024 G1025 M1026 P1028 W1029 D1116 H1119 P1120 C1122 Y1134 K1135 R1137 N1159 M1201 K1202 N1205 R1206 W1207 E8 I9 G10 M11 P13 W14 D113 H116 P117 C119 Y134 K135 R137 N157 M204 K205 N210 R211 W212 3.4.21.5 0004252,0005509,0006508,0007596 P00734 1001C~ 1014K IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4e7r G 2.25 BS02 peptide J 0 F1034 Q1038 L1065 R1067 R1073 T1074 Y1076 K1081 I1082 F19 Q24 L60 R62 R68 T69 Y71 K77 I78 3.4.21.5 0004252,0005509,0006508,0007596 P00734 1555 ~ 1565 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4e7r G 2.25 BS03 0NW G 1 H1057 Y1060A W1060D N1098 L1099 D1189 A1190 C1191 E1192 S1195 V1213 W1215 G1216 E1217 G1219 H43 Y47 W50 N95 L96 D192 A193 C194 E195 S198 V218 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 P00734 1302 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4e7r H 2.25 BS01 peptide L 0 E23 M26 P28 W29 D116 H119 P120 C122 Y134 K135 R137 N159 M201 K202 N205 R206 W207 E8 M11 P13 W14 D113 H116 P117 C119 Y134 K135 R137 N156 M203 K204 N209 R210 W211 3.4.21.5 0004252,0005509,0006508,0007596 P00734 1C~ 14K IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4e7r H 2.25 BS02 peptide I 0 F34 L40 R67 R73 T74 R75 Y76 I82 F19 L26 R62 R68 T69 R70 Y71 I78 3.4.21.5 0004252,0005509,0006508,0007596 P00734 555 ~ 565 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4e7r H 2.25 BS03 0NW H 1 H57 Y60A W60D N98 L99 D189 A190 C191 E192 S195 V213 W215 G216 G219 H43 Y47 W50 N95 L96 D191 A192 C193 E194 S197 V217 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 -logKd/Ki=7.70, Ki=0.02uM P00734 302 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG